Quốc gia: Đài Loan
Ngôn ngữ: Tiếng Trung
Nguồn: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)
ETRAVIRINE
嬌生股份有限公司 台北市中山區民生東路三段2號10樓及11樓 (30814854)
J05AG04
錠劑
主成分 (Formulation of Drug Product:) ; ETRAVIRINE (0818004000) MG
塑膠瓶裝
製 劑
須由醫師處方使用
JANSSEN-CILAG SPA VIA C. JANSSEN, B.GO SAN MICHELE, 04100 LATINA, ITALY IT
etravirine
INTELENCE與抗反轉錄病毒藥物併用,適用於曾有抗病毒藥物治療經驗,對過去的治療無效,且對NNRTI及其他抗反轉錄病毒藥物產生抗藥性之愛滋病毒HIV-1感染之成人患者。
註銷日期: 2024/05/09; 註銷理由: 許可證已逾有效期; 有效日期: 2023/06/27; 英文品名: Intelence Tablets 200mg
已註銷
2013-06-27
200 INTELENCE TABLETS 200 MG 025918 1. INTELENCE T ablets 200 mg 200 2. 200 mg Etravirine 6.1 3. 200 4. 4.1 INTELENCE NNRTI HIV-1 4.2 INTELENCE INTELENCE 200 mg 100 mg 5.2 INTELENCE INTELENCE 5.2 INTELENCE 5.2 Child-Pugh A B INTELENCE INTELENCE Child-Pugh C INTELENCE 4.4 5.2 5.2 4.3 Etravirine 4.4 HIV INTELENCE HIV INTELENCE 5.1 3 V90I A98G L100I K101E / P V106I V179D / F Y181C/ I / V G190A / S INTELENCE 5.1 Etravi ne raltegravir maraviroc 4.5 1 2 4.8 INTELENCE Stevens-Johnson Syndrome < 0.1% INTELENCE NNRTI INTELENCE INTELENCE DUET INTELENCE INTELENCE DRESS TEN 4.8 DRESS 3-6 INTELENCE INTELENCE INTELENCE 65 53 56 64 INTELENCE 55 4.2 5.2 Etravirine INTELENCE Child- Pugh C 4.2 5.2 B C B C CART HIV visceral lipomatosis 酶 PIs lipoatrophy NRTIs 4.8 HIV CART CART Pneumocystis jiroveci 4.8 HIV INTELENCE tipranavir ritonavir Etravirine 76% INTELENCE 4.5 4.5 Etravirine Etravirine CYP3A4 CYP2C9 CYP2C19 苷 酶 UDPGT glucuronidation CYP 3A4 CYP2C9 CYP2C19 Etravirine Etravirine INTELENCE CYP3A4 CYP2C9 CYP2C19 Etravirine Etravirine Etravirine Etravirine CYP3A4 INTELENCE CYP3A4 Etravirine CYP2C9 CYP2C19 P-glycoprotein INTELENCE CYP2C9 CYP2C19 P-glycoprotein Etravirine ↑ ↓ ↔ ND q.d. q.a.m. b.i.d. CI Etravirine 90% CI 1.00= 苷 苷 酶 NR TIs Didanosine 400 mg q.d. Didanosine AUC ↔ 0.99 0.79-1.25 Didanosine C min ND Didanosine C max ↔ 0.91 0.58-1.42 Etravirine AUC ↔ 1.11 0.99-1.25 Etravirine C min ↔ 1.05 0.93-1.18 Etravirine C max ↔ 1.16 1.02-1.32 Didanosine Etravirine INTELENCE didanosine Tenofovir 300 mg q.d. Tenofovir AUC ↔ 1.15 1.09-1.21 Tenofovir C min ↑ 1.19 1.13-1.26 Tenofovir C max ↑ 1.15 1.04-1.27 Etravirine AUC ↓ 0.81 0.75-0.88 Etravirine C min ↓ 0.82 0.73-0.91 Etravirine C max ↓ 0.81 0.75-0.88 Tenofovir Etravirine INTELENCE tenofovir NRTIs NRTIs abacaviremtricitabine lamivudinestavudinezidovudine INTELENCE INTELENCE NRTIs 苷 酶 NNR TIs Efavirenz Nevirapine NNRTIs INTELENCE Efavirenz Nevirapine Etravirine INTELENCE INTELENCE NNRTIs 酶 PIs ritonavir Nelfinavir INTELENCE Nelfinavir INTEL Đọc toàn bộ tài liệu