Country: Taívan
Tungumál: kínverska
Heimild: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)
TOPIRAMATE
嬌生股份有限公司 台北市中山區民生東路三段2號10樓及11樓 (30814854)
N03AX11
錠劑
TOPIRAMATE (9200038300) MG
塑膠瓶裝;;鋁箔盒裝
製 劑
須由醫師處方使用
CILAG AG. HOCHSTRASSE 201 CH-8200 SCHAFFHAUSEN SWITZERLAND CH
topiramate
用於成人及兩歲以上兒童局部癲癇或併有LENNOX-GASTAUT症候群之癲癇及原發性全身性強直陣攣癲癇的輔助治療,用於PARTIAL ONSET SEIZURE病患之單一藥物治療、預防偏頭痛。
有效日期: 2029/06/07; 英文品名: TOPAMAX FILM-COATED TABLETS 200MG
1999-06-07
® TOPAMAX ® FILM-COATED TABLETS 200 200 mg 022510 ® TOPAMAX ® FILM-COATED TABLETS 200 200 mg 022510 AED AED TOPAMAX Phenytoin Carbamazepine CBZ Valproic acid Lamotrigine Phenobarbital Primidone ↔ ** ↔ ↔ ↔ ↔ ↔ ↓ 48% ↓ 40% ↔ ↔ NS NS ↔ = < 15% ** = ↓ = NS = AED = Digoxin TOPAMAX digoxin AUC 12% digoxin TOPAMAX digoxin TOPAMAX TOPAMAX TOPAMAX 50 200 mg/day EE AUC TOPAMAX estrogen Lithium lithium topiramate 200 mg/day lithium 18% for AUC lithium topiramate 200 mg/day lithium topiramate 600 mg/day 26% for AUC topiramate lithium Risperidone topiramate 100 250 400 mg/day risperidone 1 6 mg/day steady-state AUC 250 mg/day 400 mg/day 16% 33% risperidone 9-hydroxyrisperidone 9-hydroxyrisperidone Risperidone topiramate Hydrochlorothiazide HCTZ HCTZ 25 mg 24 Topiramate 96 mg 12 HCTZ topiramate topiramate C max 27% AUC 29% HCTZ topiramate topiramate HCTZ topiramate topiramate HCTZ HCTZ topiramate Metformin metformin metformin topiramate metformin topiramate metform in topiramate metformin C max AUC 0-12h 18% 25% CL/F 20% Topiramate metformin t max Topiramate metformin metformin topiramate Metformin topiramate metformin TOPAMAX Pioglitazone topiramate pioglitazone pioglitazone AUC τ ,ss 15% C max,ss hydroxy- C max,ss AUC τ ,ss 13% 16% keto- C max,ss AUC τ ,ss 60% TOPAMAX pioglitazone pioglitazone TOPAMAX Glyburide glyburide 5 mg/day topiramate 150 mg/day Topiramate glyburide AUC 24 25% 4-trans-hydroxy-glyburide M1 3-cis-hydroxyglyburide M2 13% 15% Topiramate glyburide topiramate glyburide glyburide topiramate TOPAMAX TOPAMAX Vitamin K- topiramate vitamin K- 酶 / Prothrombin Time/International Normalized Ratio, PT/INR topiramate vitamin K- INR topiramate C max AUC topiramate topiramate topiramate a Topiramate a Amitriptyline ↔ nortriptyline C max AUC 20% NS Dihydroergotamine ↔ ↔ Haloperidol ↔ AUC 31% NS Propranolol ↔ 4-OH propranolol TPM 50 mg q12h C max 17% C max 9% 16% AUC 9% 17% 40 mg 80 mg propranolol q12h Sumatriptan ↔ NS Pizotifen ↔ ↔ Diltiazem Diltiazem AUC 25% DEA Lestu allt skjalið