×ž×“×™× ×”: טייוו×ן
שפה: ×¡×™× ×™×ª
מקור: 衛生ç¦åˆ©éƒ¨é£Ÿå“藥物管ç†ç½² (Ministry of Health and Welfare, Food And Drug Administration)
PACLITAXEL
æè¼è—¥å“å·¥æ¥è‚¡ä»½æœ‰é™å…¬å¸ 宜è˜ç¸£å†¬å±±é„‰ä¸å±±æ‘ä¸å±±è·¯84ã€84之4ã€84之6ã€84之7號ã€å†¬å±±é„‰ä¸å±±æ‘新寮路95ã€95之1ã€100之7ã€100之13ã€100之15ã€100之16ã€103ã€136號 (42042734)
L01CD01
注射劑
PACLITAXEL (1013000100) MG
注射瓶;;注射瓶;;ç›’è£
製 劑
é™ç”±é†«å¸«ä½¿ç”¨
æè¼è—¥å“å·¥æ¥è‚¡ä»½æœ‰é™å…¬å¸ 宜è˜ç¸£å†¬å±±é„‰ä¸å±±æ‘ä¸å±±è·¯ï¼˜ï¼”號 TW
paclitaxel
晚期åµå·¢ç™Œã€è…‹ä¸‹æ·‹å·´è½‰ç§»ä¹‹ä¹³ç™Œï¼Œä½œç‚ºæŽ¥çºŒå«æœè–©é¯æ¯”辛(DOXORUBICIN)在內之輔助化å¸ç™‚法ã€å·²ä½¿ç”¨åˆä½µç™‚法(除éžæœ‰ç¦å¿Œï¼Œè‡³å°‘應包括使用ANTHRACYCLINE抗癌藥)失敗的轉移乳癌ã€éžå°ç´°èƒžè‚ºç™Œã€æ„›æ»‹ç—…相關å¡æ³¢è¥¿æ°è‚‰ç˜¤ä¹‹ç¬¬äºŒç·šç™‚法;與CISPLATIN併用,作為晚期åµå·¢ç™Œä¹‹ç¬¬ä¸€ç·šç™‚法。與GEMCITABINE併用,å¯ä½¿ç”¨æ–¼æ›¾ç¶“使用éŽANTHRACYCLINE之局部復發且無法手術切除或轉移性之乳癌病患ã€èˆ‡HERCEPTIN併用時,用於治療未接å—éŽåŒ–å¸æ²»ç™‚之轉移性且乳癌éŽåº¦è¡¨ç¾HER-2之病人。
有效日期: 2026/05/24; 英文å“å: PHYXOL INJECTION 6MG/ML "SINPHAR"
2001-05-24
PIC/S GMP Paclitaxel Paclitaxel Paclitaxel taxanes Paclitaxel CAS 33069-62-4(USAN) Paclitaxel 853.929 Castor Oil Polyoxyl 35(Cremophor) Citric Acid Anhydrous Dehydrated Alcohol 2 Paclitaxel ( 300mg/m ) 3 24 (Cmax) (AUC) paclitaxel (biphasic decline) paclitaxel 2 135 175 mg/m 3 24 13.1 52.7 12.2 2 23.8 L/h/m paclitaxel 198 2 688 L/m / AUC paclitaxel (0- ) paclitaxel 89% paclitaxel Cimetidine ranitidine dexamethasone diphenhydramine paclitaxel paclitaxel P450 CYP2C8 6 - hydroxypaclitaxel CYP3A4 3 - p-hydroxypaclitaxel 6 , 3 -p-dihydroxypaclitaxel paclitaxel 6 - hydroxypaclitaxel ( ) 2 1 6 24 paclitaxel15~275 mg/m 1.3% 12.6% paclitaxel 3 225 250 2 mg/m paclitaxel 120 14 % 71% 56% 101% Paclitaxel 5% 6 - hydroxypaclitaxel paclitaxel 35 3 paclitaxel 2 2 (ULN) 175mg/m paclitaxel >2 ULN 2 (110mg/m) ( ) paclitaxel (antimicrotubule agent) (tubulin dimers) (microtubules) (reorganisation) paclitaxel Paclitaxel ( ) ( ) Paclitaxel ; Paclitaxel Ames CHO/HGPRT Paclitaxel Paclitaxel ( ) doxorubicin anthracycline CISPLATIN GEMCITABINE anthracycline Herceptin HER-2 paclitaxel polyoxyl 35 ( ) 3 Paclitaxel <1500cells/mm 3 <1000cells/mm (AIDS) ( ) Paclitaxel Paclitaxel Paclitaxel H 2 ( ) Paclitaxel Paclitaxel diphenhydramine H ( ) 2 paclitaxel paclitaxel ( ) ( ) paclitaxel 3 1500cells/mm 3 ( <1000cells/mm) paclitaxel paclitaxel 3 (<500cells/mm), 20% ( ) Paclitaxel Paclitaxel Paclitaxel Paclitaxel trastuzumab doxorubicin ( :Paclitaxel+trastuzumab Paclitaxel+doxorubicin ) Paclitaxel 20% Paclitaxel 396 mg/mL ( ) ( ) ( ) Paclitaxel+cisplatin ) O O O O O O NH OH OH OH H O O O O O 6 / Injection 6mg/mL PHYXOL ¡ Û P450 2C8 3A4 : Paclitaxel P450 CYP2C8 CYP3A4 Paclitaxel P450 CYP2C8 CYP3A4 ( :rifampicin carbamazepine phenytoin efarenz nerapine) ( :erythromycin fluoxetine gemfibrozil) paclitaxel 6 - hydroxypaclitaxel (ketoconazole verapamil diazepam quinidine dexamethasone Cyclosporine teniposide etoposide ncristine) Testosterone 17 -ethinyl estradiol retinoic acid montelukast CYP2C8 quercetin 6 - hydroxypaclitaxel Paclitaxel CYP2C8 / CYP3A4 C ×§×¨× ×ת המסמך השל×