国家: 台湾
语言: 中文
来源: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)
AMPHOTERICIN B
香港商吉立亞醫藥有限公司台灣分公司 臺北市信義區松仁路32號10樓之1、36號10樓之1 (54376860)
J02AA01
凍晶乾粉注射劑
主成分 () ; AMPHOTERICIN B (0812200102) MG
小瓶
製 劑
限由醫師使用
Gilead sciences, Inc. 1800 Wheeler Avenue, La Verne, California, 91750 USA US
amphotericin B
• 治療感染囊球菌腦膜炎的HIV患者• 治療嚴重全身性及/ 或深部黴菌感染• 治療臟器的利時曼氏病。在免疫不全且患有臟器的利時曼氏病之患者使用AmBisome治療,在初期寄生蟲清除後仍有高復發率。• 對發燒的重度嗜中性白血球缺乏症患者可能罹患黴菌感染症之經驗療法。
有效日期: 2027/03/01; 英文品名: AMBISOME FOR INJECTION
2002-03-01
AmBisome Amphotericin B, USP 50 mg hydrogenated soy phosphatidylcholine 213 mg cholesterol NF 52 mg distearoylphosphatidylglycerol 84 mg alpha tocopherol USP 0.64 mg sucrose NF 900 mg disodium succinate hexahydrate 27 mg pH 5.0 – 6.0 AmBisome Liposomal amphophilic AmBisome Amphotericin B amphophilic Amphotericin B AmBisome AmBisome 100 nm Amphotericin B Streptomyces nodosus Amphotericin B [ 1R- 1R*,3S*,5R*,6R*,9R*,11R*,15S*,16R*,17R*,18S*,19E,21E,23E,25E,27E,29E, 31E, 33R*,35S*,36R*,37S* ] -33- [ 3-Amino-3,6-dideoxy- β -D-mannopyranosyl oxy ] - 1,3,5,6,9,11,17,37-octahydroxy-15,16,18-trimethyl-13-oxo-14,39-di oxabicyclo [ 33.3.1 ] nonatriaconta-19,21,23,25,27,29,31-heptaene-36-carboxylic acid CAS No. 1397-89-3 . Amphotericin B C 47 H 73 NO 17 924.09 AmBisome Amphotericin B s t e ro l ergosterol NA + , K + , H + , and Cl - Amphotericin B ergosterol cholesterol AmBisome Amphotericin B Liposomal intracellular extracellular AmBisome Amphotericin B Aspergillus fumigatus Aspergillus flavus Candida albic ans , Candida krusei , Candida lusitaniae Candida parapsilosis , Candida tropicalis Cryptococcus neoformans Blastomyces dermatitidis 2 3 AmBisome amphotericin B Sporothrix schenckii Candida glabrata Candida krusei Candida tropicalis Candida lusitaniae Candida parapsilosis Aspergillus terreus amphotericin B AFST- EUCAST 1 2 1 AmBisome [ µg/mL ] C. albicans 59 0.015-0.12 C. glabrata 18 0.5-1 C. parapsilosis 18 0.5-1 C. krusei 19 0.5-2 C. lusitaniae 9 0.06-0.125 C. tropicalis 10 0.25-1 C. guilliermondii 4 0.06-0.12 Saccharomyces cerevisiae 3 0.03-0.06 Cryptococcus neoformans var. neoformans 10 0.06-0.12 Cryptococcus neoformans var. gattii 3 0.03-0.06 Trichosporon inkin 3 0.03-0.06 Trichosporon asahii 4 0.01-0.03 Geotrichum candidum 4 0.06-0.25 2 AmBisome [ µg/mL ] A. fumigatus 29 0.5-2 A. terreus 34 2-4 A. flavus 21 1-4 A. niger 13 1-2 * Rhizomucor species 17 0.3-0.125 Absidia corymbifera 4 0.125-1 Absidia species 17 0.5-2 Rhizopus microsporus var. oligosporus 3 0.03-0.25 Rhizopus oryzae 6 1-4 Rhizopus species 12 1-4 阅读完整的文件