Država: Tajvan
Jezik: kitajščina
Source: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)
PILOCARPINE HCL
天義企業股份有限公司 台北市復興南路一段129號5樓 (22180049)
N07AX01
錠劑
主成分 () ; PILOCARPINE HCL (5220000310) MG
瓶裝
製 劑
須由醫師處方使用
AMDIPHARM LIMITED 17 NORTHWOOD HOUSE, NORTHWOOD AVENUE, SANTRY, DUBLIN 9, IRELAND IE
pilocarpine
因頭頸部癌放射線治療造成唾腺功能減低而引起的口乾燥症。SJOGREN'S SYNDROME 所引起的口乾燥症。
有效日期: 2027/09/12; 英文品名: SALAGEN TABLETS 5MG
2002-09-12
● Pilocarpine hydrochloride 5mg ● Salagenpilocarpine hydrochlo- ridePilocarpine hydrochloride pilocarpine hydrochloride 2 ( 3 H ) - F u r a n o n e , 3 - e t h y l d i h y d r o -4-[(1-methyl-1H-imidazol-5-yl)methyl]-mono- hydrochloride, (3S-cis)244.72 S a l a g e n 5 m g pilocarpine hydrochloride Microcrystalline cellulose Stearic acid Opadry White OY-7300 Carnauba wax ● � muscarinic pilocarpine Pilocarpine M u s c a r i n i c a g o n i s t pilocarpine pilocarpine 12 5mg 10mg Salagen 20 1 3~5() 20712 Salagen 1 5mg63% 10mg90% SJOGREN’S SYNDROME12 629 Salagen 2.5~7.5mgSalagen AUC Salagen 12 () ● (8a.m.)(6p.m.)5mg 10mgpilocarpine hydrochloride 2 5mg 0.7610mg 1.35Tmax 1.250.85 Cmax15 ng/ml41 ng/ml6 AUC33ng x h/ml(5mg)108ng x h/ml(10mg) 5Cmax AUC 2 12 Salagen Tmax1.47 0.87 Cmax51.859.2ng/ml Pilocarpine Pilocarpine Pilocarpine pilocarpine acid Pilocarpine 5~25,000 ng/ml Pilocarpine (N=12) 5mg30% ( AUC) 30%2.1 ( 25.4mL/min 9.8~40.8mL/min)(N=8) Pilocarpine ● 20712(142 65) 58.5 ( 17~77)95% 4%1%Salagen tablets 5mg 10mg 16212 (14265) 57.8 ( 27~80 )88% 10%2% Salagen tablets 2.5mg 5mg10mg Salagen tablets 5 mg673 6610mg 7 4 Salagen tablets 2.5mg Salagen tablets 5 mg10 mg SJOGREN’S SYNDROME Sjogren’s Syndrom Sjogren’s Syndrom 256(14242)12 57 ( 24~85)91% 6 % 3 % Salagen tablets 5mg(20mg/) 5mg 7.5mg Salagen “ ” (visual analogue scale 100mm) 55mm 373 (16357)12 55 ( 21~84)80% 14%2%4% 2.5mg pilocarpine tablets5mg Salagen tablets 125mg 2.5mg(10mg/ ) 2.5mg(9) 5mg (16) 10~20mg/ Salagen ● Sjogren’s Syndrome ● pilocarpine ( ) ● pilocarpine pilocarpine pilocarpine pilocarpine pilocarpine pilocarpine ( ) Pilocarpine pilocarpine ● Pilocarpine Pilocarpine pilocarpine Pilocarpine ( ) agonist 5mg (Child-Pugh score of 5-6) (Child-Pugh score of 10-15) Child-Pugh *Trey, Burns, and Saunders(1966) Reference: Pugh R.N.H., Murray-Lyon, I.M., Dawson, J.L., Pietroni, M.C., Williams, R. Transection of the Oesophagus for Bleeding Oesophageal Varices, Brit. J.Surg., 1973.60:646-9 pilocarpine pilocarpine b- pilocarpine p Preberite celoten dokument