Kraj: Tajwan
Język: chiński
Źródło: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)
EPTIFIBATIDE
美商默沙東藥廠股份有限公司台灣分公司 台北市信義區信義路五段106號12樓 (86683720)
B01AC16
注射劑
EPTIFIBATIDE (9200050400) MG
小瓶;;盒裝
製 劑
限由醫師使用
PATHEON ITALIA S.P.A. VIA MOROLENSE 87, 03013 FERENTINO, ITALY IT
eptifibatide
預防不穩定性心絞痛及非Q 波心肌梗塞病人的惡化。經皮腔間冠狀動脈血管擴張術的輔助治療,以預防突發性動脈血管閉塞及相關的急性缺血併發症。
註銷日期: 2017/05/11; 註銷理由: 自請註銷; 有效日期: 2017/06/18; 英文品名: INTEGRILIN INJECTION 0.75MG/ML
已註銷
2002-06-18
2 /0.75 / INTEGRILIN IV BOLUS 2 MG/ML & IV INFUSION 0.75 MG/ML 023459 023468 Integrilin eptifibatide cysteine amide mercaptopropionyl Integrilin 10 ml2 mg/ml eptifibatide100 ml 0.75 mg/ml eptifibatide EptifibatideRGD (arginine - glycine -aspartate) Eptifibatide fibrinogen von-Willebrand GP IIb/IIIa eptifibatide ADP (adenosine diphosphate) Eptifibatide 180 mcg/ kg 2.0 mcg/kg-minADP80 %80 % 2.0 mcg/ kg-min 50 % PPACK (D-phenylalanyl-L-prolyl-L-arginine chloromethyl ketone)Qeptifibatide ADP50%(IC 50 )557 ng/ml80% (IC 80 )1100 ng/ml Integrilin 5 2-6 eptifibatide(PT)(aPTT) eptifibatide eptifibatide Integrilin Eptifibatide90-250 mcg/kg0.5-3.0 mcg/kg-min 2.0 mcg/kg-min eptifibatide 1.5-2.2 mcg/ml 180 mcg/kg Eptifibatide 25%2.555-80 ml/kg/hr185-260 ml/kg ( 74 ) / (CrCl) ( Cockcroft-Gault CrCl 50 ml/min*) ( Cockcroft-Gault CrCl 50 ml/min*) Eptifibatide(CrCl50 ml/min)50% () PURSUIT (UA) ST (NSTEMI) PURSUIT 27 726 10948 UA NSTEMI 24(10) ST ST 0.5 mm 30 ST 0.5 mm T(1 mm) CK-MB Integrilin 180 mcg/kg 2.0 mcg/kg/min (180/2.0) Integrilin 180 mcg/kg1.3 mcg/kg/min(180/1.3) (CABG) 72 PCI Integrilin2496 180/1.3 PCI CABG PURSUIT13%Integrilin(percutaneous Coronary Intervention, PCI)50%(intracoronary stent)87%(Integrilin PCI) acetylsalicylic acid (75-325 mg) (unfractionated heparin)5000 unit 1000 unit/hr aPTT 50-70 1250 72 PCIheparin(ACT)200-350 30 (MI) ( )MICK-MBQ Integrilin 180/2.0 (1)1000 15 Integrilin ( 72-96 )6 Integrilin3-4 ECG(ST) (CK-MBtroponins) ESPRIT ESPRIT (Enhanced Suppression of the Platelet IIb/IIIa Receptor with Integrilin TherapyIntegrilin IIb/IIIa ) PCI 922064PCI PCIGP IIb/IIIa 24 ( ) 90 PCI Integrilin ESPRIT Integrilin 180 mcg/kg 18-24 PERIGEE PRIDEPERIGEEPRIDE/ PERIGEE PURSUIT PRIDE PCI PERIGEE PRIDE Integrilin 2.65 μg/mL eptifibatide PCI 10 175 μmol/l 2.0 mcg/kg/min 175 350 μmol/l 1.0 mcg/kg/min0.5 mcg/kg/min 12 Integrilin ( ) Integrilin Integrilin aspirin (99.7%) 97.1% thienopyridine (95.4% clopidogel 2.7% ticlopidine) PCI 53.1% thienopyridine (52.7% clopidogel 0.5%ticlopidine)(loading dose) (30 mg) (aspirin99. Przeczytaj cały dokument