安吐平膠囊80毫克

Country: Taívan

Tungumál: kínverska

Heimild: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)

Virkt innihaldsefni:

APREPITANT

Fáanlegur frá:

萬達藥業有限公司 臺北市中山區南京東路1段52號2樓(M002)室 (50785821)

ATC númer:

A04AD12

Lyfjaform:

膠囊劑

Samsetning:

APREPITANT (9200095800) MG

Einingar í pakka:

ALU-OPA/ALU/PVC 鋁箔盒裝

Tegund:

製 劑

Gerð lyfseðils:

須由醫師處方使用

Framleitt af:

PHARMATHEN INTERNATIONAL S.A. INDUSTRIAL PARK, 5TH BLOCK, 69300, SAPES, RODOPI, GREECE GR

Lækningarsvæði:

aprepitant

Ábendingar:

與其他止吐藥劑併用,可以防止由高致吐性及中致吐性癌症化療藥物在初次或重覆使用時所引起的急性或延遲性噁心與嘔吐。

Vörulýsing:

有效日期: 2027/12/06; 英文品名: Apreto Capsules 80mg

Leyfisdagur:

2022-12-06

Upplýsingar fylgiseðill

                                安吐平膠囊
APRETO CAPSULES
(APREPITANT)
އᕥЁᝂ
$prepitant
࢚Σᆗ
substance P neurokinin 1 (NK
1
)
Ϩڱᡧࢆ״ᏢȎ
ಬԣ
ؚᘅ

ωݒጼ᠎֮
80
హքܠ
125
హք
aprepitant
ˤ
ؚᘅጼ᠎֮θӠ፷צᏢ

Hypromellose 2910, Poloxamer 407, Sucrose
和
Microcrystalline cellulose
。膠囊殼的成
分為
Gelatin, Sodium Lauryl Sulfate, Titanium dioxide
和
Black Printing Ink
,
125
毫克的
膠囊殼另含有
Iron oxide Red
色素。
ᖧסᜈ౳ᏺ
պҬᐪᚇ
Aprepitant
ژԮᑉੵީպҬዋԜȑڙᄑΫᝂ
substance P neurokinin 1(NK
1
)
ީ௯ڱᡧȌ
ژԮᒿᐏܜᇎେࡣᒛӵβީࢆ״ᏢȎဎүऄᄑᑬᒿᔸᡥݼ
(counter-screening assay)
ᡡ
Һᇎڙьሟીȍᚇႆޚ፾
(transporter)
ȍ᚞Ϗഇႈ
(ion channel)
шЏ౴աЇᕥПଞީ◩Р
ہქӯ
(Chemotherapy Induced Nausea and Vomiting
Ȍ
CINV)
ᕥݼϨዉީڱᡧѝࢌԅЛ
ἇ
(dopamine)
ᇎՠెી
(serotonin)
ީڱᡧ๓вႀϨθȌ
aprepitant
ᄑ
NK
1
ީᒿᐏܜ՗З
େ
3,000
অшκȎ
ᖧסࠓऌيᡡҺȌ
NK
1
-
ڱᡧࢆ״Ꮲѩш᙮үϥወպҬȌ؅ڣүಪवࢽܜᝂЇᕥᜈޚ
(
ڇ
ԍȒ
cisplatin)
ܤПଞީქӯȎᖧסࠓऌيᇎΫᡧҝϏ݃৬ᘨኃ௷ᆊ
(Positron Emission
Tomography, PET)
ީ๠ݘᡡҺȌ
aprepitant
ѩшघഐ໖έဨകȌٸնᐍဨകީ
NK
1
ڱ
ᡧȎᖧסࠓऌيᡡҺȌ
aprepitant
ᄑϥወًಥީպҬਬ໬ࡨߧȌѩш؅ڣ
cisplatin
Пଞ
ީࡲܜිᇎ܇ᓀිީქӯȌٸѩቲெژЯӯպҬީ
5-HT
3
-
ڱᡧࢆ״Ꮲ
ondansetron
ᇎҴ
፾ᝂۈ᎟
dexamethasone
๓ᄑ
cisplatin
ܤПଞީქӯީ؅ڣպҬȎ
ᜈ
୧ᏺ (PHARMACOKINETICS)
֦ԧ
Aprepitant
ީҋֹ๢ᄑωݒҫᡧѩҬ౯
(mean absolute oral bioavailability)
ύढࣙ
60
՗
65%
ȌՎ
aprepitant
ީҋֹീେՠϥᐲࡣ
(C
max
)
ύढј౴ӿݒᜈ
4
ϓਬ࡭
(T
max
)
Ȏ
Aprepitant
ጼ᠎ᇎዉྯԨᓫΣଞݒҬਬȌᄑ
aprepitant
ωݒҫᡧѩҬ౯ȌӿᖧסκتԮ
݌ᡡީኑ៴Ȏ
ӿᖧסᏢໞጜ൦ϻȌ
aprepitant
ީᜈޚ୧βᏺ֟౴߲ጭܜީ᜺ࠇȎ୔ீԛሐԣΫӿ༇ॿ
࡭ݒҬ
aprepitant
൚ΣᏢໞȌӿ
80 mg
՗
125 mg
Ꮲໞጜ൦Ȍڙ
AUC
0-
f
ީቲћвҬᜈ
Ꮲໞቲћвڇ
                                
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